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2,3-DIHYDRO-9H-ISOXAZOLO (3,2-B) QUINAZOLIN-9-ONES AND 3,4-DIHYDRO-(1,2)-OXAZINO (3,2-B) QUINAZOLIN-10 (2H)-ONES.REISNER DB; LUDWIG BJ; SIMON E et al.1977; ARZNEIMITTEL-FORSCH.; DTSCH.; DA. 1977; VOL. 27; NO 4; PP. 766-770; ABS. ALLEM.; BIBL. 11 REF.Article

Arylpropanolamines : Selective β3 agonists arising from strategies to mitigate phase I metabolic transformationsWASHBURN, W. N; HARPER, T. W; DEJNEKA, T et al.Bioorganic & medicinal chemistry letters (Print). 2007, Vol 17, Num 15, pp 4290-4296, issn 0960-894X, 7 p.Article

Affinity purification of endothia protease with a novel renin inhibitor, SQ 32,970NORMAN, J. A; LITTLE, D; FREE, C. A et al.Biochemical and biophysical research communications (Print). 1989, Vol 161, Num 1, pp 1-7, issn 0006-291XArticle

Quinoline-4-carboxylic acids as angiotensin II receptor antagonistsLLOYD, J; RYONO, D. E; SPITZMILLER, E. R et al.Bioorganic & medicinal chemistry letters (Print). 1994, Vol 4, Num 1, pp 195-200, issn 0960-894XArticle

(Phosphinyloxy)acyl amino inhibitors of angiotensin converting enzyme. II, Terminal amino acid analogues of (S)-1-[6-amino-2-[[hydroxy(4-phenylbutyl)phosphinyl]oxy]-1-oxohexyl]-L-prolineKARANEWSKY, D. S; BADIA, M. C; CUSHMAN, D. W et al.Journal of medicinal chemistry (Print). 1990, Vol 33, Num 5, pp 1459-1469, issn 0022-2623, 11 p.Article

Aminodiol HIV protease inhibitors. Synthesis and structure-Activity relationships of P1/P1' compounds : Correlation between lipophilicity and cytotoxicityCHEN, P; CHENG, P. T. W; JACOBS, G. A et al.Journal of medicinal chemistry (Print). 1996, Vol 39, Num 10, pp 1991-2007, issn 0022-2623Article

1,4-substituted indoles: a potent and selective class of angiotensin II receptor antagonistsPOSS, M. A; ZHENGXIANG GU; DELANEY, C. L et al.Bioorganic & medicinal chemistry letters (Print). 1994, Vol 4, Num 1, pp 145-150, issn 0960-894XArticle

β-Lactam synthesis: chemospecific sulfonation and cyclization of the β-hydroxyvaline nucleusSLUSARCHYK, W. A; DEJNEKA, T; ZAHLER, R et al.ZAHLER, R et al.Tetrahedron letters. 1986, Vol 27, Num 25, pp 2789-2792, issn 0040-4039Article

Dual metalloprotease inhibitors: Mercaptoacetyl-based fused heterocyclic dipeptide kinetics as inhibitors of angiotensin-converting enzyme and neutral endopeptidaseROBL, J. A; SUN, C.-Q; MISRA, R. N et al.Journal of medicinal chemistry (Print). 1997, Vol 40, Num 11, pp 1570-1577, issn 0022-2623Article

Orally active prodrugs of quinoline-4-carboxylic acid angiotensin II receptor antagonistsRYONO, D. E; LLOYD, J; MORELAND, S et al.Bioorganic & medicinal chemistry letters (Print). 1994, Vol 4, Num 1, pp 201-206, issn 0960-894XArticle

Diol sulfonamides : a potent and novel class of inhibitors of human reninPOSS, M. A; REID, J. A; WELLER, H. N et al.Bioorganic & medicinal chemistry letters (Print). 1993, Vol 3, Num 12, pp 2739-2744, issn 0960-894XArticle

(Phosphinyloxy)acyl amino acid inhibitors of angiotensin converting enzyme (ACE). I: Discovery of (S)-1-[6-amino-2-[[hydroxy(4-phenylbutyl)phosphinyl]oxy]-1-oxohexyl]-L-proline, a novel orally active inhibitor of ACEKARANEWSKY, D. S; BADIA, M. C; CUSHMAN, D. W et al.Journal of medicinal chemistry (Print). 1988, Vol 31, Num 1, pp 204-212, issn 0022-2623Article

Régénération du catalyseur de chloruration oxydante de l'éthylèneDEJNEKA, T. S; KIBA, YA. M; SENECHKO, M. I et al.Himičeskaâ tehnologiâ. 1986, Num 1, pp 30-31, issn 0235-3482Article

BMS-201620: a selective beta 3 agonistWASHBURN, W. N; SUN, C.-Q; MCCANN, P. J et al.Bioorganic & medicinal chemistry letters (Print). 2004, Vol 14, Num 13, pp 3525-3529, issn 0960-894X, 5 p.Article

Beta 3 agonists. Part 1 : Evolution from inception to BMS-194449WASHBURN, W. N; SHER, P. M; SUN, C. Q et al.Bioorganic & medicinal chemistry letters (Print). 2001, Vol 11, Num 23, pp 3035-3039, issn 0960-894XArticle

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